SCHEMBL8540526

SCHEMBL8540526

O=C(NC(Cn1ccnc1)c1ccc(Cl)cn1)c1ccc(-c2ccc(Cl)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 5/20 0.53
CYP51A1 Q16850 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
S1PR3 Q99500 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24240727 0.83 CYP26A1 (0.64) CYP26A1CYP51A1
SCHEMBL24240734 0.76 CYP26A1 (0.72) CYP26A1CYP51A1CYP1A2CYP3A4CYP2D6
SCHEMBL3101929 0.74 ROCK1 (0.67) CYP26A1CYP51A1
SCHEMBL8539081 0.73 ADRA2C (0.59)
SCHEMBL8536156 0.73 CYP2A6 (0.49) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8537060 0.71 ALDH1A1 (0.47) CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL8537061 0.71 ALDH1A1 (0.42) CYP26A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8536035 0.71 CYP19A1 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL24240721 0.70 CYP51A1 (0.82) CYP51A1
SCHEMBL6192902 0.69 ADRA2C (0.54) CYP51A1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683156-B1 Acylated aminoalkanimidazoles and -triazoles CIBA GEIGY AG (CH) 1998-04-01 EP disclosed
US-5622982-A ENZYME INHIBITORS; ANTIINFLAMMATORY AGENTS SANDOZ LTD. (CH) 1997-04-22 US disclosed
EP-0683156-A1 Acylated aminoalkanimidazoles and -triazoles SANDOZ LTD. (CH) 1995-11-22 EP disclosed