SCHEMBL8540558

SCHEMBL8540558

N#Cc1ccc([N+](=O)[O-])c(-c2ncc[nH]2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.46
MAPT P10636 3/20 0.42
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.40
PKM P14618 1/20 0.40
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
KAT2B Q92831 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
GSK3A P49840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536429 0.90 VCAM1 (0.50) VCAM1MAPTCYP19A1CYP11B1CYP11B2
SCHEMBL8541143 0.79 MAPK1 (0.51) MAPTMEN1KMT2ALMNAPDE4B
SCHEMBL31658933 0.79 S100A4 (0.44) MEN1KMT2ACCNB2CDK1CCNB1
SCHEMBL8541098 0.79 TDP1 (0.47) MAPTMEN1KMT2ACCNB2CDK1
SCHEMBL8542469 0.79 TSHR (0.49) MAPTMEN1KMT2ALMNACCNB2
SCHEMBL10680334 0.76 MAPT (0.39) MAPTMEN1KMT2ALMNACCNB2
SCHEMBL8539165 0.76 MAPT (0.40) VCAM1MAPTMEN1KMT2APDE4A
SCHEMBL31486076 0.76 CYP19A1 (0.45) CYP19A1CYP11B1CYP11B2HCRTR1HCRTR2
SCHEMBL1303527 0.75 CSNK1A1 (0.50) MAPTMEN1KMT2A
SCHEMBL8536034 0.74 ESR1 (0.43) MAPTMEN1KMT2ACCNB2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed