SCHEMBL8540688

SCHEMBL8540688

Cc1c(C)c2c(c(C)c1O)CCC(C)(C(=S)N1CCN(C(c3ccc(F)cc3)c3ccc(F)cc3)CC1)O2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
ACHE P22303 10/20 0.40
MAOB P27338 1/20 0.40
BCHE P06276 8/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNB1 Q02641 1/20 0.35
CACNA1C Q13936 1/20 0.35
MAPT P10636 2/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
GSTP1 P09211 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329145 0.89 PTGS1 (0.50) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8538110 0.87 TSHR (0.44) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8543897 0.86 TTPA (0.42) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8539212 0.85 CYP3A4 (0.47) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL7335483 0.80 USP2 (0.54) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL7336256 0.78 MAPT (0.46) CYP3A4TSHRACHEOPRM1MAPT
Hydrochloric Acid SCHEMBL8814353 0.77 MAPT (0.46) CYP3A4TSHRACHEOPRM1MAPT
SCHEMBL8544837 0.77 CYP3A4 (0.52) PTGS1PTGS2CYP1A2CYP3A4TSHR
Hydrochloric Acid SCHEMBL7331438 0.77 MAPT (0.45) CYP3A4TSHRACHEOPRM1MAPT
SCHEMBL9690451 0.76 TSHR (0.49) PTGS1PTGS2CYP1A2CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587499-B1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR (FR) 1998-04-29 EP disclosed
US-5395834-A Antiarthritic agents or cardiovascular disorders ADIR ET COMPAGNIE (FR) 1995-03-07 US disclosed
US-5393775-A Administering a (2-chromanyl)alkylcarboxylic acid for disorders connected with peroxidation processes ADIR ET COMPAGNIE (FR) 1995-02-28 US disclosed
EP-0587499-A1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR ET COMPAGNIE (FR) 1994-03-16 EP disclosed