SCHEMBL8540697

SCHEMBL8540697

C=CCOC(=O)c1ccnc2cccc([N+](=O)[O-])c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
ALDH1A1 P00352 4/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 1/20 0.40
EGFR P00533 1/20 0.37
SNCA P37840 1/20 0.36
KDM4E B2RXH2 4/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35
FGFR1 P11362 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
RAB9A P51151 2/20 0.34
MET P08581 1/20 0.34
ASPH Q12797 1/20 0.34
KDM8 Q8N371 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544930 0.81 ALDH1A1 (0.49) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL8545120 0.81 ALDH1A1 (0.58) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL8545932 0.77 KDM4E (0.50) ALDH1A1TSHRPOLBEGFRKDM4E
SCHEMBL30517039 0.77 KDM4E (0.50) ALDH1A1TSHRPOLBEGFRKDM4E
SCHEMBL4288671 0.77 CYP3A4 (0.68) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL8788034 0.77 CYP3A4 (0.55) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL11757412 0.76 CYP3A4 (0.58) CYP3A4ALDH1A1TSHRHSD17B10LMNA
SCHEMBL27266429 0.76 CYP3A4 (0.58) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL8788585 0.76 CYP3A4 (0.58) CYP3A4ALDH1A1TSHRHSD17B10POLB
SCHEMBL11767742 0.75 CYP3A4 (0.56) CYP3A4ALDH1A1TSHRHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0581500-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 1998-09-09 EP disclosed
US-5441949-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1995-08-15 US disclosed
EP-0581500-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-02-02 EP disclosed