SCHEMBL8540883

SCHEMBL8540883

c1ccc(OCCN2CCC(CCn3ccnc3)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 5/20 0.65
TMEM97 Q5BJF2 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
LTA4H P09960 2/20 0.54
KMT2A Q03164 1/20 0.53
NOS1 P29475 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
CACNA1B Q00975 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038254 0.92 TBXAS1 (0.55) TBXAS1TMEM97SIGMAR1LTA4HKMT2A
SCHEMBL8545842 0.81 CCR3 (0.56)
SCHEMBL8544146 0.81 GRIN2B (0.56) TBXAS1LTA4HKMT2AKDM4EALDH1A1
SCHEMBL10370478 0.80 TBXAS1 (1.00) TBXAS1LTA4HKMT2ANOS1KDM4E
SCHEMBL8538300 0.80 GRIN2B (0.54) SIGMAR1
SCHEMBL8693762 0.79 TMEM97 (0.68) TMEM97SIGMAR1LTA4HKMT2A
Hydrochloric Acid SCHEMBL9996050 0.79 TBXAS1 (0.97) TBXAS1LTA4HKMT2ANOS1KDM4E
SCHEMBL8545375 0.79 SIGMAR1 (0.59) SIGMAR1KMT2A
Hydrochloric Acid SCHEMBL8546852 0.79 GRIN2B (0.53) TBXAS1SIGMAR1
SCHEMBL8695655 0.78 TMEM97 (0.66) TMEM97SIGMAR1LTA4HKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed