SCHEMBL8543784

SCHEMBL8543784

CS(=O)(=O)O[C@@H]1C[C@@H](C(=O)N2CCN(CCO)CC2)N(C(=O)OCc2ccc([N+](=O)[O-])cc2)C1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 5/20 0.39
KCNH2 Q12809 5/20 0.39
CCR5 P51681 4/20 0.38
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
OPRK1 P41145 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8438015 1.00 KCNJ1 (0.39) KCNJ1KCNH2CCR5HRH2HRH1
SCHEMBL8438360 0.91 KCNJ1 (0.38) KCNJ1KCNH2CCR5HRH2HRH1
SCHEMBL9126331 0.88 KCNJ1 (0.39) KCNJ1KCNH2CCR5HRH2HRH1
SCHEMBL8438315 0.88 KCNJ1 (0.39) KCNJ1KCNH2CCR5HRH2HRH1
SCHEMBL8438589 0.85 KCNJ1 (0.42) KCNJ1KCNH2HRH2HRH1ALDH1A1
SCHEMBL8536750 0.85 KCNJ1 (0.42) KCNJ1KCNH2HRH2HRH1ALDH1A1
SCHEMBL9368164 0.85 ATM (0.37) KCNJ1KCNH2CCR5ALDH1A1
SCHEMBL8440034 0.85 KCNJ1 (0.41) KCNJ1KCNH2HRH2HRH1ALDH1A1
SCHEMBL9519895 0.84 TDP1 (0.42) CCR5ALDH1A1
SCHEMBL10513490 0.83 TDP1 (0.41) CCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0518558-B1 1-Methylcarbapenem derivatives, their preparation and their use as antibiotics SANKYO CO (JP) 1998-09-02 EP disclosed
EP-0518558-A1 1-Methylcarbapenem derivatives, their preparation and their use as antibiotics Sankyo Company Limited (JP) 1992-12-16 EP disclosed