SCHEMBL8543785

SCHEMBL8543785

NC(=Cc1ccc(-c2ccccc2)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.52
WDR5 P61964 1/20 0.47
POLB P06746 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
EGFR P00533 1/20 0.43
CA1 P00915 1/20 0.42
MGLL Q99685 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CYP3A4 P08684 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TAAR1 Q96RJ0 1/20 0.39
MMP3 P08254 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8543781 1.00 TP53 (0.52) TP53WDR5POLBMEN1KMT2A
SCHEMBL911941 0.87 AKR1C1 (0.50) POLBMEN1KMT2APRSS1PRSS2
SCHEMBL1567874 0.87 AKR1C1 (0.50) POLBMEN1KMT2APRSS1PRSS2
SCHEMBL12449789 0.87 AKR1C1 (0.50) POLBMEN1KMT2APRSS1PRSS2
SCHEMBL13485353 0.82 ESR1 (0.54) TP53POLBMEN1KMT2ANPC1
SCHEMBL8543155 0.82 MAOB (0.49) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL8550468 0.82 PTGS2 (0.49) POLBMEN1KMT2AEGFRNPC1
SCHEMBL8550464 0.82 PTGS2 (0.49) POLBMEN1KMT2AEGFRNPC1
SCHEMBL8543162 0.82 MAOB (0.49) MEN1KMT2AEGFRNPC1RAB9A
SCHEMBL338880 0.78 CYP19A1 (0.61) TP53POLBMEN1KMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0671385-B1 Method for handling (2-alkyl) acryloyl isocyanate, method for producing (2-alkyl)acryloyl isocyanate, heterocyclic compound, and method for producing heterocyclic compound NIPPON PAINT CO LTD (JP) 1998-10-14 EP disclosed
US-5663423-A Method for handling (2-alkyl) (acryloyl) isocyanate, method for stabilizing (2-alkyl) (acryloyl) isocyanate, method for producing (2-alkyl) (acryloyl) isocyanate, heterocyclic compound, and method for producing heterocyclic compound NIPPON PAINT CO., LTD (JP) 1997-09-02 US disclosed
US-5532360-A REACTING WITH AZOMETHINE COMPOUND TO FORM HETEROCYCLIC COMPOUND NIPPON PAINT CO., LTD. (JP) 1996-07-02 US disclosed
EP-0671385-A1 Method for handling (2-alkyl) acryloyl isocyanate, method for producing (2-alkyl)acryloyl isocyanate, heterocyclic compound, and method for producing heterocyclic compound Nippon Paint Co., Ltd. (JP) 1995-09-13 EP disclosed