SCHEMBL8550464

SCHEMBL8550464

Cc1ccc(/C=C(/N)c2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.49
MAPT P10636 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
CYP3A4 P08684 1/20 0.49
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
POLB P06746 1/20 0.45
EGFR P00533 1/20 0.44
CYP2D6 P10635 1/20 0.43
HIF1A Q16665 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CYP1B1 Q16678 1/20 0.41
GRIN2D O15399 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550468 1.00 PTGS2 (0.49) PTGS2MAPTALDH1A1HPGDCYP3A4
SCHEMBL9398625 0.90 PTGS2 (0.46) PTGS2MAPTALDH1A1HPGDCES2
SCHEMBL12449789 0.85 AKR1C1 (0.50) MAPTALDH1A1HPGDCYP3A4POLB
SCHEMBL911941 0.85 AKR1C1 (0.50) MAPTALDH1A1HPGDCYP3A4POLB
SCHEMBL1567874 0.85 AKR1C1 (0.50) MAPTALDH1A1HPGDCYP3A4POLB
SCHEMBL8543785 0.82 TP53 (0.52) PTGS2MAPTCYP3A4NPC1RAB9A
SCHEMBL8543781 0.82 TP53 (0.52) PTGS2MAPTCYP3A4NPC1RAB9A
SCHEMBL8543155 0.80 MAOB (0.49) PTGS2MAPTALDH1A1CYP3A4CES2
SCHEMBL8543162 0.80 MAOB (0.49) PTGS2MAPTALDH1A1CYP3A4CES2
SCHEMBL15460561 0.79 ALDH1A1 (0.40) PTGS2MAPTALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262025-A2 Organic electroluminescent device TDK Corporation (JP) 2010-12-15 EP disclosed
EP-0671385-B1 Method for handling (2-alkyl) acryloyl isocyanate, method for producing (2-alkyl)acryloyl isocyanate, heterocyclic compound, and method for producing heterocyclic compound NIPPON PAINT CO LTD (JP) 1998-10-14 EP disclosed
US-5663423-A Method for handling (2-alkyl) (acryloyl) isocyanate, method for stabilizing (2-alkyl) (acryloyl) isocyanate, method for producing (2-alkyl) (acryloyl) isocyanate, heterocyclic compound, and method for producing heterocyclic compound NIPPON PAINT CO., LTD (JP) 1997-09-02 US disclosed
US-5532360-A REACTING WITH AZOMETHINE COMPOUND TO FORM HETEROCYCLIC COMPOUND NIPPON PAINT CO., LTD. (JP) 1996-07-02 US disclosed
EP-0671385-A1 Method for handling (2-alkyl) acryloyl isocyanate, method for producing (2-alkyl)acryloyl isocyanate, heterocyclic compound, and method for producing heterocyclic compound Nippon Paint Co., Ltd. (JP) 1995-09-13 EP disclosed