SCHEMBL8544444

SCHEMBL8544444

O=C(C1CCc2[nH]cnc2C1)N1CC(c2ccccc2O)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
IDH1 O75874 11/20 0.39
ADRA1A P35348 4/20 0.37
HTR3A P46098 2/20 0.37
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
SLC6A4 P31645 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
KCNH2 Q12809 1/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
ADRA1D P25100 1/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8538933 0.99 KDM4E (0.39) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
SCHEMBL8544447 0.92 HTR3A (0.45) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
Hydrochloric Acid SCHEMBL8538937 0.91 HTR3A (0.44) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
SCHEMBL8479741 0.89 ADRA1A (0.40) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
SCHEMBL8538941 0.88 IDH1 (0.38) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
Hydrochloric Acid SCHEMBL8538095 0.88 ADRA1A (0.40) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
Hydrochloric Acid SCHEMBL8539594 0.87 IDH1 (0.37) KDM4ESMN1; SMN2IDH1ADRA1AHTR3A
SCHEMBL8525220 0.86 IDH1 (0.36) IDH1ADRA1AHTR3AADRA2AADRA2B
SCHEMBL8540938 0.85 IDH1 (0.37) KDM4EIDH1ADRA1AHTR3AADRA2A
Hydrochloric Acid SCHEMBL8540899 0.85 IDH1 (0.35) IDH1ADRA1AHTR3AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721949-B1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE CO (JP) 1998-01-07 EP claimed
US-5677326-A GASTROINTESTINAL DISORDERS TOKYO TANABE COMPANY LIMITED (JP) 1997-10-14 US claimed
EP-0721949-A1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE COMPANY LIMITED (JP) 1996-07-17 EP claimed
EP-0721949-B1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE CO (JP) 1998-01-07 EP disclosed
US-5677326-A GASTROINTESTINAL DISORDERS TOKYO TANABE COMPANY LIMITED (JP) 1997-10-14 US disclosed
EP-0721949-A1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE COMPANY LIMITED (JP) 1996-07-17 EP disclosed