SCHEMBL8544673

SCHEMBL8544673

CC(=O)NC(=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.72

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.72
HPGD P15428 1/20 0.72
KMT2A Q03164 5/20 0.65
MEN1 O00255 4/20 0.65
CES2 O00748 1/20 0.62
CES1 P23141 1/20 0.62
TP53 P04637 1/20 0.60
POLB P06746 2/20 0.59
MAPT P10636 2/20 0.59
BLM P54132 1/20 0.59
CRHBP P24387 1/20 0.59
CRHR2 Q13324 1/20 0.59
TSHR P16473 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
GAA P10253 2/20 0.58
ATM Q13315 1/20 0.58
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060904 0.90 KMT2A (0.73) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL10355 0.87 KMT2A (0.69) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL4603889 0.86 ALDH1A1 (0.75) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL11068063 0.85 KMT2A (0.74) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL6995692 0.85 KMT2A (0.67) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL24933536 0.84 ALDH1A1 (0.64) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL11064012 0.83 CYP1A2 (0.70) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL8298069 0.82 ALDH1A1 (0.70) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL29508878 0.81 KMT2A (0.71) ALDH1A1HPGDKMT2AMEN1CES2
SCHEMBL297043 0.81 KMT2A (0.71) ALDH1A1HPGDKMT2AMEN1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508796-B1 Cholecystokinin antagonists MERCK & CO INC (US) 1998-07-08 EP disclosed
US-5220018-A Benzodiazepine derivatives MERCK & CO., INC. (US) 1993-06-15 US disclosed
EP-0508796-A1 Cholecystokinin antagonists MERCK & CO. INC. (US) 1992-10-14 EP disclosed
US-4447515-A DIACYLAMINE COMPOUND ADDED FUJI PHOTO FILM CO., LTD. (JP) 1984-05-08 US disclosed