SCHEMBL8544834

SCHEMBL8544834

COc1cc(OC)c(C(=O)CBr)cc1OC

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
KMT2A Q03164 2/20 0.53
HPGDS O60760 1/20 0.53
HMGCR P04035 1/20 0.50
LCK P06239 1/20 0.48
FYN P06241 1/20 0.48
PAX8 Q06710 1/20 0.47
MEN1 O00255 1/20 0.47
HTT P42858 1/20 0.46
GSK3B P49841 1/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10891861 0.89 KDM4E (0.51) CYP3A4KMT2AHPGDSHMGCRLCK
SCHEMBL20508037 0.87 HPGDS (0.49) CYP3A4KMT2AHPGDSHMGCRLCK
SCHEMBL20507907 0.85 HPGDS (0.47) CYP3A4KMT2AHPGDSMEN1ALDH1A1
SCHEMBL14525270 0.85 HPGDS (0.47) CYP3A4KMT2AHPGDSHMGCRPAX8
SCHEMBL15680284 0.85 LCK (0.65) CYP3A4KMT2AHPGDSHMGCRLCK
SCHEMBL7460397 0.83 CYP3A4 (0.59) CYP3A4KMT2AHMGCRLCKFYN
SCHEMBL23173662 0.83 HPGDS (0.49) CYP3A4HPGDSHTTGSK3BALDH1A1
SCHEMBL6928976 0.83 HPGDS (0.49) CYP3A4KMT2AHPGDSHMGCRLCK
SCHEMBL4764754 0.82 HMGCR (0.72) CYP3A4KMT2AHMGCRLCKFYN
SCHEMBL679852 0.82 CYP3A4 (0.62) CYP3A4KMT2AHMGCRLCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed