SCHEMBL8544913

SCHEMBL8544913

COc1ccccc1C1(O)CCC(c2ccccc2)(c2ccccc2)C2CNCC21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.56
SIGMAR1 Q99720 1/20 0.48
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
OPRM1 P35372 3/20 0.39
OPRD1 P41143 3/20 0.39
OPRK1 P41145 3/20 0.39
OPRL1 P41146 3/20 0.39
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
FNTA P49354 2/20 0.36
FNTB P49356 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9241561 0.99 TACR1 (0.55) TACR1SIGMAR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL7886015 0.99 TACR1 (0.55) TACR1SIGMAR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8956731 0.99 TACR1 (0.55) TACR1SIGMAR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8874914 0.83 SIGMAR1 (0.49) TACR1SIGMAR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8956780 0.82 TACR1 (0.38) TACR1OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL9242986 0.81 TACR1 (0.43) TACR1SIGMAR1OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL9242969 0.81 TACR1 (0.43) TACR1SIGMAR1OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL8956811 0.81 TACR1 (0.43) TACR1SIGMAR1OPRM1OPRD1OPRK1
SCHEMBL8874681 0.80 SIGMAR1 (0.46) TACR1SIGMAR1CHRM2CHRM4CHRM5
SCHEMBL9281012 0.80 SIGMAR1 (0.43) TACR1SIGMAR1CHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635002-B1 NOVEL PERHYDROISOINDOLE DERIVATIVES AND PREPARATION THEREOF RHONE POULENC RORER SA (FR) 1998-07-22 EP claimed
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US claimed
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US disclosed