SCHEMBL9281012

SCHEMBL9281012

COc1ccccc1C1(O)C(O)CC(c2ccccc2)(c2ccccc2)[C@H]2CNCC21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
TACR1 P25103 2/20 0.40
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
KMT2A Q03164 1/20 0.36
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 2/20 0.35
OPRL1 P41146 2/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
GRIN2B Q13224 1/20 0.34
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8543227 1.00 SIGMAR1 (0.43) SIGMAR1TACR1CHRM2CHRM4CHRM5
SCHEMBL8956750 1.00 SIGMAR1 (0.43) SIGMAR1TACR1CHRM2CHRM4CHRM5
SCHEMBL8893688 1.00 SIGMAR1 (0.43) SIGMAR1TACR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8895671 0.99 SIGMAR1 (0.42) SIGMAR1TACR1CHRM2CHRM4CHRM5
SCHEMBL8875107 0.87 SIGMAR1 (0.42) SIGMAR1TACR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8893607 0.87 ALOX5AP (0.35) SIGMAR1TACR1KMT2AHTR2CHTR2B
SCHEMBL8874747 0.84 SIGMAR1 (0.46) SIGMAR1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL8956868 0.80 MAOB (0.36) HTR2AHTR2CHTR2B
SCHEMBL8544913 0.80 TACR1 (0.56) SIGMAR1TACR1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL7886015 0.79 TACR1 (0.55) SIGMAR1TACR1CHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US disclosed