SCHEMBL8544937

SCHEMBL8544937

O=C1Nc2ccc(C(O)CN3CCCC(Cc4ccccc4)C3)cc2CO1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 8/20 0.51
GRIN2D O15399 1/20 0.51
GRIN3B O60391 1/20 0.51
GRIN1 Q05586 1/20 0.51
GRIN2A Q12879 1/20 0.51
GRIN2C Q14957 1/20 0.51
GRIN3A Q8TCU5 1/20 0.51
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TBXA2R P21731 1/20 0.42
HRH1 P35367 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.40
ATM Q13315 1/20 0.40
KCNH2 Q12809 1/20 0.40
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544941 1.00 GRIN2B (0.51) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8543097 1.00 GRIN2B (0.51) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8547979 0.85 GRIN2B (0.62) GRIN2BMEN1KMT2AKDM4EALDH1A1
SCHEMBL8541679 0.85 GRIN2B (0.62) GRIN2BMEN1KMT2AKDM4EALDH1A1
SCHEMBL8547850 0.85 GRIN2B (0.62) GRIN2BMEN1KMT2AKDM4EALDH1A1
SCHEMBL8540531 0.85 GRIN2B (0.62) GRIN2BMEN1KMT2AKDM4EALDH1A1
SCHEMBL8544371 0.85 GRIN2B (0.47) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8547693 0.85 GRIN2B (0.47) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8548698 0.85 GRIN2B (0.47) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8547346 0.84 GRIN1 (0.51) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed