SCHEMBL8545014

SCHEMBL8545014

Cc1cn(CCC2CCN(C(=O)CCc3ccccc3)CC2)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPB1 P15086 2/20 0.60
GRIN2B Q13224 1/20 0.53
FAAH O00519 1/20 0.52
POLB P06746 2/20 0.52
NPC1 O15118 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
CHRM3 P20309 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
FKBP1A P62942 1/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545153 0.82 KDM4C (0.51) FAAHL3MBTL1MEN1KMT2AKDM4C
SCHEMBL8544549 0.81 GRIN2B (0.53) CPB1GRIN2BFAAHPOLBNPC1
SCHEMBL8540312 0.81 GRIN2B (0.55) CPB1GRIN2BFAAHPOLBNPC1
SCHEMBL8699576 0.81 NPC1 (0.53) CPB1GRIN2BNPC1TDP1CHRM3
SCHEMBL8540740 0.80 HRH3 (0.53) GRIN2B
SCHEMBL8545115 0.79 POLB (0.52) CPB1GRIN2BFAAHPOLBNPC1
SCHEMBL8546968 0.79 F10 (0.57) CPB1GRIN2BFAAHPOLBNPC1
SCHEMBL8544779 0.78 GRIN2B (0.60) CPB1GRIN2BFAAHPOLBNPC1
SCHEMBL9031203 0.77 POLB (0.52) GRIN2BFAAHPOLBNPC1TDP1
SCHEMBL8542324 0.77 HTT (0.58) CPB1GRIN2BFAAHPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed