SCHEMBL8540312

SCHEMBL8540312

O=C(CCc1ccccc1)N1CCC(CCn2ccnc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.55
FAAH O00519 1/20 0.54
POLB P06746 1/20 0.54
CPB1 P15086 1/20 0.53
NPC1 O15118 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
FKBP1A P62942 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
TSHR P16473 1/20 0.46
TBXAS1 P24557 1/20 0.45
CHRM3 P20309 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538696 0.94 FAAH (0.50) GRIN2BFAAHPOLBCPB1ALDH1A1
SCHEMBL8541116 0.94 FAAH (0.57) GRIN2BFAAHPOLBCPB1NPC1
SCHEMBL9031024 0.90 PKM (0.53) GRIN2BFAAHPOLBCPB1NPC1
SCHEMBL8545661 0.89 GRIN2B (0.46) GRIN2BFAAHCPB1ALDH1A1TBXAS1
SCHEMBL8540403 0.89 TBXAS1 (0.46) GRIN2BFAAHCPB1TBXAS1
SCHEMBL8541801 0.89 GRIN2B (0.57) GRIN2BFAAHPOLBNPC1TDP1
SCHEMBL8545335 0.89 HDAC3 (0.54) GRIN2BFAAHPOLBALDH1A1KDM4E
SCHEMBL8546276 0.87 CPB1 (0.55) GRIN2BPOLBCPB1NPC1TDP1
SCHEMBL8540293 0.86 CPB1 (0.44) GRIN2BFAAHPOLBCPB1TBXAS1
SCHEMBL8540305 0.86 FKBP1A (0.52) CPB1TDP1FKBP1AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed