SCHEMBL8544779

SCHEMBL8544779

O=C(CCc1ccccc1)N1CCC(CCn2nccn2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.60
POLB P06746 2/20 0.59
FAAH O00519 1/20 0.58
NPC1 O15118 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
CHRNB2 P17787 1/20 0.53
CHRNB4 P30926 1/20 0.53
CHRNA3 P32297 1/20 0.53
CHRNA4 P43681 1/20 0.53
FKBP1A P62942 1/20 0.51
ALDH1A1 P00352 2/20 0.50
TSHR P16473 1/20 0.50
NAAA Q02083 1/20 0.50
KDM4E B2RXH2 1/20 0.50
CPB1 P15086 1/20 0.49
CHRM3 P20309 1/20 0.48
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539022 0.86 POLB (0.54) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8540505 0.82 POLB (0.68) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8540312 0.81 GRIN2B (0.55) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8546036 0.81 POLB (0.54) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8546597 0.81 FAAH (0.57) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8541896 0.81 FAAH (0.56) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8541862 0.81 POLB (0.66) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8546968 0.80 F10 (0.57) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8542093 0.80 POLB (0.64) GRIN2BPOLBFAAHNPC1TDP1
SCHEMBL8541372 0.80 HDAC3 (0.56) FAAHHPGDHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed