SCHEMBL8545018

SCHEMBL8545018

N#Cc1c(Cl)ncc(C=O)c1-c1cccs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.41
MAPT P10636 5/20 0.41
HSD17B10 Q99714 3/20 0.41
POLB P06746 1/20 0.41
ALOX15 P16050 1/20 0.41
KDM4E B2RXH2 11/20 0.40
ALDH1A1 P00352 9/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
LMNA P02545 3/20 0.39
HTT P42858 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
GAA P10253 4/20 0.38
HPGD P15428 3/20 0.38
GLA P06280 1/20 0.38
CASP1 P29466 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PKM P14618 1/20 0.38
NPSR1 Q6W5P4 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548916 0.81 ALDH1A1 (0.44) ADORA1HSD17B10ALOX15KDM4EALDH1A1
SCHEMBL8544979 0.72 KMT2A (0.34) MAPTPOLBKDM4EALDH1A1MEN1
SCHEMBL31111404 0.72 KMT2A (0.34) MAPTPOLBKDM4EALDH1A1MEN1
SCHEMBL6254233 0.65 ALDH1A1 (0.68) ADORA1MAPTHSD17B10KDM4EALDH1A1
SCHEMBL10551506 0.64 ERN1 (0.45) MAPTHSD17B10KDM4EALDH1A1MEN1
SCHEMBL17795920 0.63 MAPT (0.50) ADORA1MAPTHSD17B10POLBALOX15
SCHEMBL845698 0.63 AXL (0.37) ADORA1ALDH1A1KMT2ANPSR1ADORA2A
SCHEMBL1028588 0.62 MAPT (0.45) ADORA1MAPTHSD17B10POLBALOX15
SCHEMBL12679799 0.62 KDM4E (0.55) ADORA1MAPTHSD17B10POLBALOX15
SCHEMBL7395814 0.62 ERN1 (0.43) ADORA1MAPTHSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702003-B1 Process for preparing 2-halogenpyridinaldehydes BAYER AG (DE) 1998-06-17 EP disclosed
US-5708180-A CYCLIZATION OF UNSATURATED NITRILE, AMIDE OR OXIME BAYER AKTIENGESELLSCHAFT (DE) 1998-01-13 US disclosed
EP-0702003-A2 Process for preparing 2-halogenpyridinaldehydes and new 2-halogenpyridinaldehydes BAYER AG (DE) 1996-03-20 EP disclosed