SCHEMBL8545117

SCHEMBL8545117

CCOC(=O)c1cc2c(N3CCN(CCc4ccc(Cl)cc4)CC3)cccc2s1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 14/20 0.53
SLC6A4 P31645 2/20 0.53
DRD2 P14416 11/20 0.46
HTR2A P28223 10/20 0.46
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44
KCNJ1 P48048 1/20 0.44
KCNH2 Q12809 1/20 0.44
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
DRD4 P21917 1/20 0.42
SMYD2 Q9NRG4 1/20 0.42
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8546533 0.99 HTR1A (0.52) HTR1ASLC6A4DRD2HTR2AHTR1D
SCHEMBL8545233 0.93 HTR1A (0.54) HTR1ASLC6A4DRD2HTR2AHTR1D
Hydrochloric Acid SCHEMBL8545102 0.92 HTR1A (0.53) HTR1ASLC6A4DRD2HTR2AHTR1D
SCHEMBL8545047 0.92 HTR1A (0.53) HTR1ASLC6A4DRD2HTR2AHTR1D
SCHEMBL8549120 0.91 HTR1A (0.53) HTR1ASLC6A4DRD2HTR2AHTR1D
Hydrochloric Acid SCHEMBL8545546 0.91 HTR1A (0.52) HTR1ASLC6A4DRD2HTR2AHTR1D
SCHEMBL8551141 0.90 ADRA1D (0.52) HTR1ASLC6A4DRD2HTR2AHTR1D
Hydrochloric Acid SCHEMBL8543418 0.90 HTR1A (0.52) HTR1ASLC6A4DRD2HTR2AHTR1D
Hydrochloric Acid SCHEMBL8549073 0.89 ADRA1D (0.52) HTR1ASLC6A4DRD2HTR2AHTR1D
SCHEMBL8544023 0.88 HTR1A (0.48) HTR1ASLC6A4DRD2HTR2AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed