SCHEMBL8545310

SCHEMBL8545310

Cc1ccc(S(=O)(=O)NC(=O)CC(=O)O)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.60
ERBB2 P04626 4/20 0.60
LMNA P02545 3/20 0.57
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
MMP1 P03956 1/20 0.55
MMP2 P08253 1/20 0.55
MMP9 P14780 1/20 0.55
MMP8 P22894 1/20 0.55
MMP13 P45452 1/20 0.55
ALDH1A1 P00352 4/20 0.54
KMT2A Q03164 2/20 0.54
RAB9A P51151 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
ALB P02768 1/20 0.54
CYP2C9 P11712 1/20 0.54
TSHR P16473 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
POLB P06746 1/20 0.53
PTGS2 P35354 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6279910 0.88 EGFR (0.56) EGFRERBB2LMNACA1CA2
SCHEMBL28405273 0.85 EGFR (0.60) EGFRERBB2LMNACA1CA2
SCHEMBL7969578 0.85 EGFR (0.60) EGFRERBB2LMNACA1CA2
SCHEMBL692083 0.84 LMNA (0.64) LMNACA1CA2MMP1MMP2
SCHEMBL13537908 0.84 CA1 (0.68) EGFRERBB2LMNACA1CA2
SCHEMBL2635660 0.84 EGFR (0.63) EGFRERBB2LMNACA1CA2
SCHEMBL5931139 0.84 ALDH1A1 (0.71) EGFRERBB2LMNACA1CA2
SCHEMBL5177119 0.83 EGFR (0.55) EGFRERBB2LMNACA1CA2
SCHEMBL13800951 0.82 EGFR (0.51) EGFRERBB2LMNAALDH1A1KMT2A
Ammonia Solution, Strong SCHEMBL6098128 0.82 LMNA (0.62) LMNACA1CA2MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580633-B1 HETEROCYCLIC AMINES USEFUL IN THE THERAPY OF ASTHMA AND INFLAMMATION OF THE RESPIRATORY TRACT BOEHRINGER MANNHEIM ITALIA (IT) 1998-06-17 EP disclosed
US-5453423-A Heterocyclic amines useful in the therapy of asthma and imflammation of the respiratory tract BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1995-09-26 US disclosed
EP-0580633-A1 HETEROCYCLIC AMINES USEFUL IN THE THERAPY OF ASTHMA AND INFLAMMATION OF THE RESPIRATORY TRACT BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1994-02-02 EP disclosed
WO-1992018478-A1 HETEROCYCLIC AMINES USEFUL IN THE THERAPY OF ASTHMA AND INFLAMMATION OF THE RESPIRATORY TRACT BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-10-29 WO disclosed