SCHEMBL8545345

SCHEMBL8545345

O=C(O)c1c(-c2ccccc2)c2cc(OCc3ccccc3)ccc2n1Cc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 10/20 0.69
EDNRA P25101 9/20 0.69
SERPINE1 P05121 5/20 0.54
PLA2G2A P14555 1/20 0.48
S1PR5 Q9H228 1/20 0.47
MAPK8 P45983 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856902 0.91 EDNRB (0.58) EDNRBEDNRASERPINE1S1PR5MAPK8
SCHEMBL4711435 0.84 MAPK8 (0.66) EDNRBEDNRAMAPK8
SCHEMBL8540948 0.83 EDNRA (0.72) EDNRBEDNRAS1PR5
SCHEMBL6858271 0.81 EDNRB (0.55) EDNRBEDNRAPLA2G2A
SCHEMBL8551430 0.81 EDNRB (0.80) EDNRBEDNRASERPINE1PLA2G2A
SCHEMBL8643680 0.81 EDNRA (0.78) EDNRBEDNRA
SCHEMBL6858334 0.80 EDNRB (0.62) EDNRBEDNRASERPINE1PLA2G2A
SCHEMBL8856638 0.80 EDNRA (0.78) EDNRBEDNRA
SCHEMBL8857076 0.80 EDNRB (0.64) EDNRBEDNRA
SCHEMBL8856815 0.79 EDNRB (0.74) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800389-A4 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 1998-04-29 EP claimed
EP-0800389-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1997-10-15 EP claimed
WO-1996018393-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1996-06-20 WO claimed
US-5684032-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC, ANTIASTHMATIC AGENTS AND RESPIRATORY DISORDERS SMITHKLINE BEECHAM CORPORATION (US) 1997-11-04 US disclosed