SCHEMBL8545474

SCHEMBL8545474

COc1cccc(-c2cc(-c3ccc(F)cc3)nn2C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.52
ALDH1A3 P47895 2/20 0.51
SQOR Q9Y6N5 1/20 0.47
PIK3CA P42336 2/20 0.45
PIK3CG P48736 1/20 0.45
BRD4 O60885 1/20 0.45
PTGS2 P35354 1/20 0.44
NPY5R Q15761 1/20 0.43
FYN P06241 2/20 0.42
TP53 P04637 1/20 0.42
EGLN2 Q96KS0 1/20 0.42
STAT3 P40763 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
DYRK1A Q13627 1/20 0.41
NFE2L2 Q16236 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20239626 0.89 TDP1 (0.48) MAPTBRD4FYNTP53EGLN2
SCHEMBL5598135 0.86 STAT3 (0.47) MAPTPTGS2FYNSTAT3L3MBTL1
SCHEMBL17372934 0.81 MAPT (0.53) MAPTL3MBTL1MAPK1HSD17B10
SCHEMBL5597739 0.79 BACE1 (0.46) MAPTFYNTP53STAT3L3MBTL1
SCHEMBL6693299 0.78 ATM (0.55) MAPTPTGS2STAT3DYRK1AMAPK1
SCHEMBL14458205 0.77 MAPT (0.46) MAPTTP53EGLN2L3MBTL1MAPK1
SCHEMBL24314980 0.76 ALDH1A3 (0.58) MAPTALDH1A3SQORBRD4NPY5R
SCHEMBL30610970 0.76 ALDH1A3 (0.58) MAPTALDH1A3SQORBRD4NPY5R
SCHEMBL5597719 0.75 ESR2 (0.54) MAPTFYNHSD17B10
SCHEMBL5385380 0.75 GABRG2 (0.51) NPY5REGLN2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1092186-C Preparation method of 1, 2-dimethyl-3, 5-diaryl pyrazolium methylsulfate BASF AG (DE) 2002-10-09 CN disclosed
US-5847154-A Method of preparing 1,2-dimethyl-3,5-diarylpyrazolium methylsulfates BASF AKTIENGESELLSCHAFT (DE) 1998-12-08 US disclosed
CN-1192734-A Preparation method of 1, 2-dimethyl-3, 5-diaryl pyrazolium methylsulfate BASF AG (DE) 1998-09-09 CN disclosed