SCHEMBL8545486

SCHEMBL8545486

Nc1c2c(nc3ccccc13)CCc1cn(Cc3ccccc3)nc1-2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ACHE P22303 8/20 0.45
BCHE P06276 7/20 0.45
HTR2C P28335 1/20 0.43
ADORA3 P0DMS8 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CACNB4 O00305 1/20 0.42
CACNA1A O00555 1/20 0.42
SLC22A2 O15244 1/20 0.42
SLC22A1 O15245 1/20 0.42
ABCC4 O15439 1/20 0.42
CACNA1G O43497 1/20 0.42
CACNG3 O60359 1/20 0.42
CACNA1F O60840 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549310 0.89 ADORA2A (0.44) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8544321 0.87 BCHE (0.46) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8545346 0.85 BCHE (0.44) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8543400 0.84 BCHE (0.44) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8543857 0.84 ACHE (0.44) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8547014 0.84 ACHE (0.44) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8545134 0.84 KDM4E (0.50) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8545799 0.83 ACHE (0.43) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8544712 0.83 ACHE (0.49) MEN1KMT2AACHEBCHEADORA3
SCHEMBL8545791 0.82 IGF1R (0.42) ACHEBCHEADORA3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5179100-A Analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-01-12 US claimed
EP-0560231-B1 Pyrazolo(3,4-a)acridine derivatives as analgesics HOECHST MARION ROUSSEL INC (US) 1998-06-03 EP disclosed
EP-0560231-A1 Pyrazolo(3,4-a)acridine derivatives as analgesics HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-09-15 EP disclosed
US-5179100-A Analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-01-12 US disclosed