SCHEMBL8546353

SCHEMBL8546353

CC(C)(C)OC(=O)N[C@@H](c1ccc(F)cc1F)[C@@H](O)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.41
CTSK P43235 3/20 0.41
KDM4D Q6B0I6 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
AAK1 Q2M2I8 2/20 0.39
PPARG P37231 3/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
NCOA2 Q15596 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
TRPA1 O75762 1/20 0.38
PTPN1 P18031 1/20 0.37
ACE P12821 1/20 0.37
S1PR3 Q99500 1/20 0.36
GABRB1 P18505 1/20 0.35
GABRB2 P47870 1/20 0.35
PPARA Q07869 3/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8741363 0.89 KDM4D (0.39) CTSSCTSKKDM4DCES2CES1
SCHEMBL4177618 0.85 CTSS (0.46) CTSSCTSKPPARGPTPN1ACE
SCHEMBL29571131 0.83 CTSS (0.43) CTSSCTSKKDM4DCES2CES1
SCHEMBL3822263 0.83 CTSS (0.43) CTSSCTSKKDM4DCES2CES1
SCHEMBL6439819 0.82 CTSS (0.46) CTSSCTSKAAK1PPARGLMNA
SCHEMBL17041588 0.80 TRPA1 (0.44) CTSSCTSKKDM4DCES2CES1
SCHEMBL8912111 0.80 CTSS (0.47) CTSSCTSKCES2CES1PPARG
SCHEMBL30765251 0.78 CTSS (0.43) CTSSCTSKCES2CES1AAK1
SCHEMBL3762203 0.78 CTSS (0.43) CTSSCTSKCES2CES1AAK1
SCHEMBL16680101 0.78 CTSA (0.45) CTSSCTSKKDM4DTSHRJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0693485-B1 Baccatin derivatives and processes for preparing the same TANABE SEIYAKU CO (JP) 1998-06-03 EP disclosed
US-5677470-A CHEMICAL INTERMEDIATES; ANTITUMOR AGENTS TANABE SEIYAKU CO., LTD. (JP) 1997-10-14 US disclosed
EP-0693485-A2 Baccatin derivatives and processes for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1996-01-24 EP disclosed