SCHEMBL8546355

SCHEMBL8546355

CC(C)(CCOc1ccc(CNO)cc1)CCOc1ccc(CNO)cc1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
PDE4A P27815 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HIF1A Q16665 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
THRB P10828 1/20 0.39
IDO1 P14902 1/20 0.39
TSHR P16473 1/20 0.39
MITF O75030 1/20 0.39
GAA P10253 1/20 0.39
CYP3A4 P08684 1/20 0.39
EPHX2 P34913 1/20 0.38
NR1H4 Q96RI1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551864 0.83 THRB (0.50) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8544675 0.81 THRB (0.48) ALDH1A1KDM4ECYP1A2CYP2D6PDE4A
SCHEMBL8543274 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8551450 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8549440 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8544062 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8550526 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8552037 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL8551534 0.80 S1PR2 (0.47) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL6254887 0.74 CYP3A4 (0.46) ALDH1A1KDM4ESMN1; SMN2GAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed