SCHEMBL8546409

SCHEMBL8546409

CON=C(C)Cn1nnn(C(=O)N(c2ccccc2)C(C)C)c1=O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.38
LMNA P02545 2/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
TRPM8 Q7Z2W7 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
USP2 O75604 1/20 0.32
MLYCD O95822 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
ATM Q13315 1/20 0.31
PKM P14618 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546039 0.85 ALDH1A1 (0.43) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL8550089 0.83 ALDH1A1 (0.42) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL9620371 0.80 ALDH1A1 (0.46) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL8546014 0.80 ALDH1A1 (0.41) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL8346740 0.78 ALDH1A1 (0.43) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL9620447 0.78 ALDH1A1 (0.43) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL8690403 0.77 ALDH1A1 (0.49) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL8550504 0.77 ALDH1A1 (0.43) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL7977970 0.76 ALDH1A1 (0.42) ALDH1A1LMNATP53SMN1; SMN2MEN1
SCHEMBL9620586 0.76 ALDH1A1 (0.42) ALDH1A1LMNATP53SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed
EP-0820994-A1 Tetrazolinones as herbicides and intermediates NIHON BAYER AGROCHEM K.K. (JP) 1998-01-28 EP disclosed