SCHEMBL8547645

SCHEMBL8547645

NC1(F)C=CC=CC1C(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.38
NPC1 O15118 1/20 0.38
CES1 P23141 3/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
ALOX15 P16050 1/20 0.35
HBB P68871 1/20 0.35
TSHR P16473 2/20 0.34
CYP2C19 P33261 2/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 1/20 0.34
PARP1 P09874 1/20 0.34
RECQL P46063 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
EPHX1 P07099 2/20 0.34
CES2 O00748 2/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7851780 0.85 L3MBTL1 (0.41) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL6938598 0.82 L3MBTL1 (0.39) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL8989984 0.81 CES1 (0.41) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL5564543 0.81 L3MBTL1 (0.38) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL1828048 0.78 L3MBTL1 (0.41) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL7782761 0.77 L3MBTL1 (0.36) L3MBTL1NPC1MAPTHTTALOX15
SCHEMBL3165913 0.77
SCHEMBL4621722 0.77 NPC1 (0.40) L3MBTL1NPC1CES1MAPTHTT
SCHEMBL28014454 0.75 NPC1 (0.42) L3MBTL1NPC1CES1MAPTHTT
Hydrazine SCHEMBL28754327 0.75 NPC1 (0.37) L3MBTL1NPC1CES1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508796-B1 Cholecystokinin antagonists MERCK & CO INC (US) 1998-07-08 EP disclosed
US-5220018-A Benzodiazepine derivatives MERCK & CO., INC. (US) 1993-06-15 US disclosed
EP-0508796-A1 Cholecystokinin antagonists MERCK & CO. INC. (US) 1992-10-14 EP disclosed
US-4628084-A AMIDATION, AMMONIATION, CONDENSATION MERCK & CO., INC. (US) 1986-12-09 US disclosed