SCHEMBL8547747

SCHEMBL8547747

O=C1CCc2cc(C(=O)CCN3CCC[C@H](Cc4ccccc4)C3)ccc2N1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.54
HTR1A P08908 2/20 0.50
HTR2A P28223 2/20 0.50
HTR7 P34969 2/20 0.50
DRD3 P35462 2/20 0.50
DRD4 P21917 1/20 0.50
ACHE P22303 3/20 0.47
OGT O15294 1/20 0.47
DRD2 P14416 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
CARM1 Q86X55 1/20 0.44
PRMT6 Q96LA8 1/20 0.44
CRBN Q96SW2 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547953 1.00 GRIN2B (0.54) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8547562 0.95 ACHE (0.49) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8871868 0.93 GRIN2B (0.54) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8549788 0.93 GRIN2B (0.54) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8548011 0.91 GRIN2B (0.62) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8542972 0.89 GRIN2B (0.60) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8547760 0.86 GRIN2B (0.47) GRIN2BACHECARM1PRMT6
SCHEMBL8549221 0.86 GRIN2B (0.57) GRIN2BACHEOGTCRBN
SCHEMBL8545426 0.86 GRIN2B (0.57) GRIN2BACHEOGTCRBN
SCHEMBL8549819 0.85 GRIN2B (0.58) GRIN2BHTR1AHTR2AHTR7DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed