SCHEMBL8548407

SCHEMBL8548407

CC1(C)CC(=O)Nc2c(Cl)cc(C(O)CCN3CCC[C@H](Cc4ccccc4)C3)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 2/20 0.43
PRMT6 Q96LA8 2/20 0.43
GRIN2B Q13224 4/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
BCHE P06276 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
HTR2A P28223 2/20 0.38
CCR3 P51677 2/20 0.38
CCR2 P41597 2/20 0.37
CHRNB2 P17787 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8591795 1.00 CARM1 (0.43) CARM1PRMT6GRIN2BGRIN2DGRIN3B
SCHEMBL8544988 0.93 MEN1 (0.41) CARM1PRMT6GRIN2BBCHECCR3
SCHEMBL8544991 0.93 MEN1 (0.41) CARM1PRMT6GRIN2BBCHECCR3
SCHEMBL8543130 0.93 MEN1 (0.41) CARM1PRMT6GRIN2BBCHECCR3
SCHEMBL8541668 0.91 GRIN2B (0.51) GRIN2BGRIN2DGRIN3BADRA1DADRA1A
SCHEMBL8591796 0.88 CARM1 (0.43) CARM1PRMT6GRIN2BGRIN2DGRIN3B
SCHEMBL8548411 0.88 CARM1 (0.43) CARM1PRMT6GRIN2BGRIN2DGRIN3B
SCHEMBL8873521 0.84 CARM1 (0.43) CARM1PRMT6GRIN2BBCHEHTR2A
SCHEMBL8542893 0.84 CARM1 (0.43) CARM1PRMT6GRIN2BBCHEHTR2A
SCHEMBL8542815 0.82 ALDH1A1 (0.42) CARM1PRMT6HTR2ACCR3CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed