Malonic Acid

Malonic Acid

SCHEMBL8548541

COc1cccc(N(C(N)=S)c2ccc3oc(C)c(CCN(C)CCc4ccncc4)c3c2)c1.O=C(O)CC(=O)O

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.35
TP53 P04637 5/20 0.35
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 5/20 0.34
RAB9A P51151 3/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 1/20 0.34
NR3C2 P08235 1/20 0.34
MTNR1A P48039 6/20 0.34
MTNR1B P49286 6/20 0.34
NPC1 O15118 2/20 0.33
POLB P06746 1/20 0.33
KDM4C Q9H3R0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Malonic Acid SCHEMBL8549235 0.95 MAPT (0.36) MAPTTP53KDM4EMEN1CYP1A2
Malonic Acid SCHEMBL7147604 0.85 KDM4E (0.44) MAPTKDM4EMEN1KMT2ASMN1; SMN2
Malonic Acid SCHEMBL8552650 0.85 SMN1; SMN2 (0.34) MAPTTP53KDM4ECYP1A2CYP3A4
Malonic Acid SCHEMBL7146355 0.80 HTR1D (0.43) MAPTKDM4EMEN1KMT2ASMN1; SMN2
Malonic Acid SCHEMBL8550508 0.80 SMN1; SMN2 (0.35) MAPTKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8552137 0.76 GNRHR (0.34) MAPTTP53KDM4EKMT2ASMN1; SMN2
SCHEMBL8549069 0.75 GNRHR (0.38) MAPTTP53KDM4EMEN1CYP1A2
SCHEMBL28382188 0.60 PARP1 (0.56) TP53MTNR1AMTNR1BHTT
SCHEMBL10669106 0.60 NPSR1 (0.49) MAPTTP53KDM4EMEN1CYP1A2
SCHEMBL7144826 0.59 MAPT (0.45) MAPTKDM4EMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed