SCHEMBL8548880

SCHEMBL8548880

O=C(Oc1ccccc1C(=O)CN1CCC[C@H]1C(=O)NCc1ccccc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
PTGER4 P35408 2/20 0.49
F2 P00734 4/20 0.49
FKBP1A P62942 2/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPSR1 Q6W5P4 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC3 O15379 1/20 0.46
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548313 0.87 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2PTGER4FKBP1ACYP3A4
SCHEMBL8548877 0.86 NPSR1 (0.43) ALDH1A1SMN1; SMN2CYP2C9CYP2C19NPSR1
SCHEMBL8548878 0.86 NPSR1 (0.43) ALDH1A1SMN1; SMN2CYP2C9CYP2C19NPSR1
SCHEMBL8548111 0.86 ALDH1A1 (0.52) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A
SCHEMBL8548491 0.85 PTGER4 (0.52) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A
SCHEMBL8543317 0.84 F2 (0.58) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A
SCHEMBL8545355 0.83 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A
SCHEMBL8545367 0.82 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2FKBP1ACYP3A4CYP2C9
SCHEMBL8545019 0.79 F2 (0.56) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A
SCHEMBL8544635 0.79 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2PTGER4F2FKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed