SCHEMBL8549392

SCHEMBL8549392

CCCCCN1CCC(c2csc3ccc(NC(=S)Nc4ccc(-c5ccccc5)cc4)cc23)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.50
SLC6A4 P31645 1/20 0.50
CHRM3 P20309 7/20 0.39
BCHE P06276 1/20 0.38
CCR2 P41597 2/20 0.37
KCNH2 Q12809 2/20 0.37
HTR3A P46098 1/20 0.37
MCHR1 Q99705 1/20 0.36
HTR1A P08908 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8708757 0.93 DRD2 (0.53) DRD2SLC6A4BCHE
SCHEMBL8550206 0.86 DRD2 (0.47) DRD2SLC6A4
SCHEMBL8702974 0.86 DRD2 (0.53) DRD2SLC6A4BCHECCR2KCNH2
SCHEMBL8549396 0.85 DRD2 (0.49) DRD2SLC6A4BCHEKCNH2HTR1A
SCHEMBL8551116 0.84 DRD2 (0.47) DRD2SLC6A4
SCHEMBL8703019 0.84 DRD2 (0.53) DRD2SLC6A4BCHECCR2
SCHEMBL7484437 0.82 HTR1D (0.55) DRD2CCR2HTR1A
SCHEMBL8548017 0.82 DRD2 (0.50) DRD2SLC6A4DRD3
SCHEMBL8706839 0.81 DRD2 (0.48) DRD2SLC6A4CHRM3CCR2KCNH2
SCHEMBL8704937 0.81 DRD2 (0.44) DRD2SLC6A4KCNH2HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed