SCHEMBL8549472

SCHEMBL8549472

CS(=O)(=O)c1ccc(N2CCN(CCNC(=O)c3ccc4c(c3)CCOC4)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.49
POLB P06746 1/20 0.48
DRD4 P21917 6/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA9 Q16790 1/20 0.46
HSD17B10 Q99714 1/20 0.46
DRD2 P14416 3/20 0.46
DRD3 P35462 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
PMP22 Q01453 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548777 0.88 HTR1D (0.54) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8553219 0.88 HTR1A (0.52) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8550457 0.87 HTR1A (0.51) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8551190 0.87 HTR1A (0.64) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8549853 0.86 DRD4 (0.65) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8549479 0.86 HTR1A (0.50) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8552310 0.85 HTR1A (0.48) HTR1APOLBDRD4HSD17B10DRD2
SCHEMBL8554330 0.84 CD274 (0.59) HTR1ADRD4DRD2DRD3
SCHEMBL8551554 0.83 DRD4 (0.46) HTR1ADRD4CA12CA1CA9
SCHEMBL8549399 0.81 CCR3 (0.56) HTR1ADRD4DRD2DRD3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed