SCHEMBL8551190

SCHEMBL8551190

O=C(NCCN1CCN(c2ccccc2)CC1)c1ccc2c(c1)CCOC2

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.64
MAPT P10636 1/20 0.60
DRD3 P35462 3/20 0.59
DRD4 P21917 2/20 0.59
DRD2 P14416 2/20 0.59
POLB P06746 1/20 0.59
HSD17B10 Q99714 1/20 0.59
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C19 P33261 1/20 0.54
HPGD P15428 1/20 0.54
CD274 Q9NZQ7 1/20 0.54
ALDH1A1 P00352 1/20 0.52
HTT P42858 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553219 0.91 HTR1A (0.52) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8548777 0.89 HTR1D (0.54) HTR1ADRD4DRD2POLBHSD17B10
SCHEMBL8549799 0.89 HTR1A (0.53) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8550457 0.88 HTR1A (0.51) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8549853 0.88 DRD4 (0.65) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8549479 0.88 HTR1A (0.50) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8554330 0.88 CD274 (0.59) HTR1ADRD3DRD4DRD2CD274
SCHEMBL8549757 0.87 DRD3 (0.59) HTR1AMAPTDRD3DRD2POLB
SCHEMBL8549472 0.87 HTR1A (0.49) HTR1AMAPTDRD3DRD4DRD2
SCHEMBL8552310 0.86 HTR1A (0.48) HTR1AMAPTDRD3DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed