SCHEMBL854978

SCHEMBL854978

O=C1OCc2cccc(Cl)c21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
TYMS P04818 1/20 0.44
CYP1A2 P05177 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 2/20 0.43
AHR P35869 1/20 0.40
CES1 P23141 1/20 0.37
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13151881 0.78 MAOA (0.32) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL9273526 0.76 PBRM1 (0.41) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL8791015 0.76 PBRM1 (0.41) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL32672790 0.75 TDP2 (0.50) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL855553 0.75 MAOA (0.47) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL1611599 0.75 MAOA (0.47) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL855947 0.75 MAOB (0.47) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL31616856 0.75 KDM4E (0.47) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL4455687 0.75 KDM4E (0.47) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL29838115 0.75 MAOA (0.47) MAOAMAOBKDM4EALDH1A1TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022204150-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CNS DISORDERS BLUE OAK PHARMACEUTICALS, INC. (US) 2022-09-29 WO disclosed
US-9309250-B2 Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-04-12 US disclosed
CN-102046580-B Methods for preparing oxydiphthalic anhydrides SABIC INNOVATIVE PLASTICS IP 2015-02-04 CN disclosed
EP-2723746-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Inc. (US) 2014-04-30 EP disclosed
US-8604221-B2 Production method of halogen-substituted phthalide SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2013-12-10 US disclosed
EP-2271611-B1 METHOD FOR PREPARING 4,4'-OXYDIPHTHALIC ANHYDRIDE SABIC INNOVATIVE PLASTICS IP (NL) 2013-09-04 EP disclosed
US-20130034616-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-02-07 US disclosed
WO-2012178125-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-12-27 WO disclosed
US-20120142946-A1 PRODUCTION METHOD OF HALOGEN-SUBSTITUTED PHTHALIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-06-07 US disclosed
EP-2433933-A1 PRODUCTION METHOD OF HALOGEN-SUBSTITUTED PHTHALIDE Sumitomo Chemical Company, Limited (JP) 2012-03-28 EP disclosed
EP-1390339-A2 PROCESS FOR THE PREPARATION OF 7-SUBSTITUTED 3-ALKYL-3H-ISOBENZOFURAN-1-ONE DERIVATIVES Syngenta Participations AG (CH) 2004-02-25 EP disclosed
EP-1375468-A2 Method for removing impurities from oxidation products GENERAL ELECTRIC COMPANY (US) 2004-01-02 EP disclosed
US-6670487-B1 Of ortho-dimethylbenzene compounds; phthalic acid and phthalic anhydride by oxidation of ortho-xylene; extracting solution of aromatic anhydride product with an aqueous bicarbonate to hydrolyze the anhydride to the acid GENERAL ELECTRIC COMPANY 2003-12-30 US disclosed
WO-2002094760-A2 PROCESS FOR THE PREPARATION OF 7-SUBSTITUTED 3-ALKYL-3H-ISOBENZOFURAN-1-ONE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2002-11-28 WO disclosed
EP-0461079-B1 Substituted phthalides and heterocyclic phthalides CIBA GEIGY AG (CH) 1997-07-16 EP disclosed
US-5627138-A HERBICIDES SANDOZ LTD. (CH) 1997-05-06 US disclosed
US-5627137-A HERBICIDES SANDOZ LTD. (CH) 1997-05-06 US disclosed
US-5561101-A HERBICIDES SANDOZ LTD. (CH) 1996-10-01 US disclosed
US-5506192-A HERBICIDES SANDOZ LTD. 1996-04-09 US disclosed
EP-0461079-A2 Substituted phthalides and heterocyclic phthalides SANDOZ LTD. (CH) 1991-12-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130034616-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, MAP3K5 MAOA 3499/4885MAOB 3227/4885KDM4E 1959/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.