SCHEMBL8549836

SCHEMBL8549836

ONCc1ccc(Sc2ccc(CNO)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.54
IDO1 P14902 1/20 0.54
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
NR1H2 P55055 1/20 0.42
PTPRZ1 P23471 2/20 0.39
PTPN1 P18031 1/20 0.39
PTGIR P43119 1/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
MITF O75030 1/20 0.36
XBP1 P17861 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NOD2 Q9HC29 1/20 0.36
HTT P42858 1/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
SLC6A4 P31645 4/20 0.35
MEN1 O00255 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6895044 0.74 THRB (0.59) THRBIDO1NOS1NOS2TSHR
SCHEMBL17065246 0.74 THRB (0.59) THRBIDO1NOS1NOS2RAB9A
SCHEMBL12447265 0.73 THRB (0.42) THRBIDO1NR1H2RAB9ANPC1
Hydrochloric Acid SCHEMBL17065240 0.72 THRB (0.56) THRBIDO1NOS1NOS2RAB9A
SCHEMBL6979704 0.72 IDO1 (0.56) THRBIDO1NOS1NOS2RAB9A
SCHEMBL4941612 0.72 THRB (0.56) THRBIDO1NOS1NOS2HTT
SCHEMBL12976226 0.72 THRB (0.56) THRBIDO1NOS1NOS2TSHR
SCHEMBL1505831 0.72 MEN1 (0.58) THRBIDO1NOS1NOS2MEN1
SCHEMBL131948 0.72 IDO1 (0.56) THRBIDO1NOS1NOS2CYP3A4
SCHEMBL7754741 0.72 THRB (0.56) THRBIDO1NOS1NOS2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed