SCHEMBL8550138

SCHEMBL8550138

CCCNC(=O)c1ccc(N2CCN(CCN(C)C(=O)c3ccc4c(c3)CCOC4)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.44
CHRNA10 Q9GZZ6 1/20 0.43
CHRNA9 Q9UGM1 1/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
DRD2 P14416 2/20 0.42
DRD3 P35462 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
NAMPT P43490 1/20 0.41
SLC2A1 P11166 1/20 0.41
HTR1A P08908 1/20 0.41
CYP1A2 P05177 1/20 0.40
PRKD1 Q15139 1/20 0.40
HTR1D P28221 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549100 0.87 DRD4 (0.47) DRD4DRD2HTR1AHTR1D
SCHEMBL8550036 0.87 DRD4 (0.47) DRD4DRD2HTR1AHTR1D
SCHEMBL8553551 0.87 DRD4 (0.48) DRD4CHRNA10CHRNA9DRD2HTR1A
SCHEMBL8550687 0.87 DRD4 (0.48) DRD4DRD2HTR1AHTR1D
SCHEMBL8551575 0.87 DRD4 (0.48) DRD4DRD2HTR1ACYP1A2HTR1D
SCHEMBL8549471 0.87 DRD4 (0.48) DRD4DRD2DRD3HTR1AHTR1D
SCHEMBL8550252 0.86 DRD4 (0.59) DRD4DRD2DRD3SLC2A1HTR1A
SCHEMBL8549843 0.85 DRD4 (0.46) DRD4DRD2DRD3HTR1AHTR1D
SCHEMBL8549485 0.85 DRD4 (0.48) DRD4DRD2HTR1AHTR1D
SCHEMBL8549415 0.84 DRD4 (0.49) DRD4DRD2HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed