SCHEMBL8549843

SCHEMBL8549843

CN(CCN1CCN(c2ccc(C(F)(F)F)cc2)CC1)C(=O)c1ccc2c(c1)CCOC2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.46
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
DRD2 P14416 4/20 0.41
AKR1C3 P42330 1/20 0.41
TACR1 P25103 1/20 0.40
TACR3 P29371 1/20 0.40
CD274 Q9NZQ7 1/20 0.39
PPARD Q03181 3/20 0.39
PPARA Q07869 3/20 0.39
DRD3 P35462 1/20 0.38
SLC6A4 P31645 1/20 0.38
RORC P51449 1/20 0.38
HTR1D P28221 4/20 0.38
HTR2A P28223 3/20 0.38
HTR1A P08908 2/20 0.38
CETP P11597 1/20 0.38
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550849 0.91 DRD4 (0.46) DRD4LMNAMAPTDRD2TACR1
SCHEMBL8549507 0.91 HTR7 (0.45) DRD4MAPTDRD2DRD3HTR2A
SCHEMBL8551575 0.89 DRD4 (0.48) DRD4DRD2HTR1DHTR2AHTR1A
SCHEMBL8553551 0.89 DRD4 (0.48) DRD4DRD2SLC6A4HTR1DHTR2A
SCHEMBL8549471 0.89 DRD4 (0.48) DRD4MAPTDRD2DRD3HTR1D
SCHEMBL8550687 0.89 DRD4 (0.48) DRD4MAPTDRD2HTR1DHTR2A
SCHEMBL8550263 0.89 DRD4 (0.48) DRD4DRD2PPARDPPARASLC6A4
SCHEMBL8550252 0.88 DRD4 (0.59) DRD4DRD2DRD3HTR2AHTR1A
SCHEMBL8549100 0.87 DRD4 (0.47) DRD4MAPTDRD2HTR1DHTR2A
SCHEMBL8550036 0.87 DRD4 (0.47) DRD4LMNAMAPTDRD2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed