SCHEMBL8550161

SCHEMBL8550161

CC[C@H](C)[C@@H](C=Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
CTSK P43235 11/20 0.47
PPARA Q07869 3/20 0.45
PPARG P37231 2/20 0.45
CTSS P25774 2/20 0.43
SYK P43405 1/20 0.42
ATM Q13315 1/20 0.42
IDO1 P14902 1/20 0.42
ACE P12821 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550157 1.00 TDP1 (0.50) TDP1CTSKPPARAPPARGCTSS
SCHEMBL8613012 1.00 TDP1 (0.50) TDP1CTSKPPARAPPARGCTSS
SCHEMBL8550164 1.00 TDP1 (0.50) TDP1CTSKPPARAPPARGCTSS
SCHEMBL8136411 0.89 CTSK (0.46) TDP1CTSKPPARAPPARGCTSS
SCHEMBL8136416 0.89 CTSK (0.46) TDP1CTSKPPARAPPARGCTSS
SCHEMBL13986003 0.82 TDP1 (0.47) TDP1CTSKPPARAPPARGCTSS
SCHEMBL10980321 0.81 PPARA (0.47) TDP1CTSKPPARAPPARGCTSS
SCHEMBL9058208 0.81 PPARA (0.47) TDP1CTSKPPARAPPARGCTSS
SCHEMBL10973888 0.81 PPARA (0.47) TDP1CTSKPPARAPPARGCTSS
SCHEMBL13986019 0.80 TDP1 (0.45) TDP1CTSKPPARAPPARGCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
EP-0610745-A2 Novel aminomethylene derivatives as immunosuppressants Bayer Corporation (US) 1994-08-17 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed