SCHEMBL8550320

SCHEMBL8550320

COC(=O)c1c(C(=O)c2ccccc2)cccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.47
NR1H3 Q13133 1/20 0.47
TSHR P16473 1/20 0.46
KCNK3 O14649 2/20 0.46
KCNK9 Q9NPC2 2/20 0.46
TAS2R14 Q9NYV8 2/20 0.44
SLC6A3 Q01959 1/20 0.43
LMNA P02545 2/20 0.43
GAA P10253 1/20 0.43
RBP4 P02753 1/20 0.42
MYC P01106 1/20 0.42
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
NOTUM Q6P988 1/20 0.41
ELANE P08246 1/20 0.41
AKR1C3 P42330 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550050 0.89 TDP1 (0.46) NR1H2KCNK3KCNK9TAS2R14LMNA
SCHEMBL8553845 0.89 CYP1A2 (0.46) NR1H2TSHRSLC6A3LMNAGAA
SCHEMBL27484659 0.84 NR1H2 (0.50) NR1H2NR1H3KCNK3KCNK9TAS2R14
SCHEMBL7041350 0.82 TSHR (0.55) TSHRSLC6A3LMNAGAAMYC
SCHEMBL1994212 0.81 CA12 (0.55) TSHRTAS2R14LMNAGAARBP4
SCHEMBL7212456 0.79 TSHR (0.52) TSHRKCNK3KCNK9SLC6A3LMNA
SCHEMBL8550492 0.79 CYP1A2 (0.44) TSHRSLC6A3GAAPDK2CA12
SCHEMBL3717986 0.78 GAA (0.56) NR1H2NR1H3KCNK3KCNK9LMNA
SCHEMBL31369140 0.78 GAA (0.56) NR1H2NR1H3KCNK3KCNK9LMNA
SCHEMBL8547750 0.78 MAPT (0.59) TSHRSLC6A3LMNAGAAMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed