SCHEMBL8553845

SCHEMBL8553845

COC(=O)c1c(C(=O)c2ccc(F)cc2)cccc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAB9A P51151 4/20 0.44
KMT2A Q03164 4/20 0.44
NPC1 O15118 3/20 0.44
MEN1 O00255 2/20 0.44
MAPT P10636 2/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
NOTUM Q6P988 1/20 0.43
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ATM Q13315 1/20 0.40
EPHX2 P34913 1/20 0.39
PDK2 Q15119 1/20 0.39
CA12 O43570 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550492 0.90 CYP1A2 (0.44) CYP1A2CYP2D6TSHRCYP2C19RAB9A
SCHEMBL8550050 0.89 TDP1 (0.46) RAB9AKMT2AMEN1MAPTNOTUM
SCHEMBL8550320 0.89 NR1H2 (0.47) TSHRKMT2AMEN1HTTSLC6A3
SCHEMBL21253254 0.84 CYP1A2 (0.55) CYP1A2CYP2D6TSHRCYP2C19RAB9A
SCHEMBL8551130 0.81 CYP1A2 (0.51) CYP1A2CYP2D6TSHRCYP2C19RAB9A
SCHEMBL8551443 0.81 ALDH1A1 (0.49) CYP1A2CYP2D6TSHRCYP2C19RAB9A
SCHEMBL8551927 0.81 CYP1A2 (0.48) CYP1A2CYP2D6TSHRCYP2C19RAB9A
SCHEMBL1994212 0.79 CA12 (0.55) TSHRNOTUMGAACA12CA1
SCHEMBL1407421 0.78 HDAC8 (0.45) GAASMN1; SMN2NR1H2LMNA
SCHEMBL8549684 0.76 ALDH1A1 (0.49) CYP1A2CYP2D6TSHRCYP2C19RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed