SCHEMBL8550446

SCHEMBL8550446

COC(=O)c1c(C#N)cccc1C(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
KDM5A P29375 1/20 0.46
SLC6A3 Q01959 1/20 0.43
ALDH1A1 P00352 5/20 0.42
NPSR1 Q6W5P4 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
NFKB1 P19838 1/20 0.42
CYP2C19 P33261 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
HIF1A Q16665 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 3/20 0.42
HSD17B10 Q99714 1/20 0.42
MYC P01106 1/20 0.42
AKR1C3 P42330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2383149 0.85 CA12 (0.48) TSHRKDM5AALDH1A1CYP1A2CYP3A4
SCHEMBL7041350 0.82 TSHR (0.55) TSHRSLC6A3ALDH1A1NPSR1CYP1A2
SCHEMBL7212456 0.79 TSHR (0.52) TSHRSLC6A3ALDH1A1NPSR1CYP1A2
SCHEMBL11756627 0.78 SMN1; SMN2 (0.50) TSHRSLC6A3ALDH1A1TDP1KDM4E
SCHEMBL14037057 0.78 TSHR (0.53) TSHRALDH1A1NPSR1CYP1A2CYP3A4
SCHEMBL1200740 0.78 AKR1C3 (0.55) ALDH1A1NPSR1MAPTTDP1AKR1C3
SCHEMBL8549312 0.78 TSHR (0.50) TSHRSLC6A3ALDH1A1NPSR1CYP1A2
SCHEMBL8547750 0.78 MAPT (0.59) TSHRSLC6A3ALDH1A1MAPTKDM4E
SCHEMBL27532725 0.77 AKR1C3 (0.47) TSHRALDH1A1NPSR1MAPTTDP1
SCHEMBL181067 0.76 ALDH1A1 (0.55) TSHRALDH1A1MAPTKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed