Bromide

Bromide

SCHEMBL8551577

Br.Cc1cc2c(cc1O)C(C1(c3cccs3)CC1)N(C)CC2

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.39
DRD1 P21728 7/20 0.39
MAOA P21397 1/20 0.39
DRD4 P21917 2/20 0.38
DRD5 P21918 1/20 0.38
DRD3 P35462 1/20 0.37
NR1I2 O75469 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420090 0.99 DRD2 (0.40) DRD2DRD1MAOADRD4DRD5
SCHEMBL7417594 0.83 MAOA (0.41) DRD2DRD1MAOADRD4MAPK1
Bromide SCHEMBL8543859 0.81 DRD2 (0.39) DRD2DRD1MAOADRD4DRD3
SCHEMBL7416842 0.80 DRD1 (0.40) DRD2DRD1MAOADRD4DRD3
Hydrochloric Acid SCHEMBL7422696 0.79 DRD2 (0.39) DRD2DRD1MAOADRD4DRD3
Bromide SCHEMBL8747087 0.78 DRD1 (0.46) DRD2DRD1MAOADRD4DRD5
SCHEMBL7473332 0.76 DRD2 (0.40) DRD2DRD1MAOADRD4DRD5
SCHEMBL8747024 0.76 DRD1 (0.47) DRD2DRD1MAOADRD4DRD5
Oxalic Acid SCHEMBL7414373 0.76 DRD1 (0.37) DRD2DRD1MAOADRD3
SCHEMBL7419696 0.76 DRD1 (0.39) DRD2DRD1MAOADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807868-A ANALGESICS; PSYCHOLOGICAL DISORDES; PARKINSON*S DIESASE;COGNITION ACTIVATORS; DRUG DEPENDENCE; DYSKINESIA KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-15 US disclosed
US-5804586-A ANALGESICS, PSYCHOLOGICAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-09-08 US disclosed
EP-0707570-B1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1998-05-06 EP disclosed