SCHEMBL8551671

SCHEMBL8551671

Cc1ccc(C(=O)OC2CCN(Cc3cccc(F)c3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.55
SCN2A Q99250 1/20 0.55
SCN3A Q9NY46 1/20 0.55
KMT2A Q03164 2/20 0.55
SIGMAR1 Q99720 5/20 0.53
TMEM97 Q5BJF2 1/20 0.53
HTR2A P28223 1/20 0.50
CCR3 P51677 1/20 0.48
CACNA1G O43497 1/20 0.48
POLB P06746 1/20 0.48
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8551715 0.99 KMT2A (0.57) SCN1ASCN2ASCN3AKMT2ASIGMAR1
SCHEMBL8551850 0.90 SIGMAR1 (0.60) KMT2ASIGMAR1CCR3
Hydrochloric Acid SCHEMBL8550732 0.89 KMT2A (0.60) KMT2ASIGMAR1CCR3
SCHEMBL8551160 0.87 SCN1A (0.61) SCN1ASCN2ASCN3AHTR2A
SCHEMBL8551873 0.87 SCN1A (0.55) SCN1ASCN2ASCN3AKMT2A
SCHEMBL8550697 0.87 SCN1A (0.55) SCN1ASCN2ASCN3AKMT2ASIGMAR1
SCHEMBL8552204 0.87 SCN1A (0.55) SCN1ASCN2ASCN3AKMT2ASIGMAR1
Hydrochloric Acid SCHEMBL8554961 0.86 SCN1A (0.60) SCN1ASCN2ASCN3AHTR2A
SCHEMBL8550662 0.86 SCN1A (0.63) SCN1ASCN2ASCN3AKMT2APOLB
Hydrochloric Acid SCHEMBL8551263 0.86 SCN1A (0.54) SCN1ASCN2ASCN3AKMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed