SCHEMBL8551160

SCHEMBL8551160

Cc1ccc(C(=O)OC2CCN(Cc3ccc(F)cc3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.61
SCN2A Q99250 1/20 0.61
SCN3A Q9NY46 1/20 0.61
ADRB2 P07550 1/20 0.56
MCHR1 Q99705 1/20 0.54
HTR2A P28223 1/20 0.53
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8554961 0.99 SCN1A (0.60) SCN1ASCN2ASCN3AADRB2MCHR1
SCHEMBL8551183 0.95 SCN1A (0.68) SCN1ASCN2ASCN3AADRB2KDM4E
Hydrochloric Acid SCHEMBL8553929 0.94 SCN1A (0.66) SCN1ASCN2ASCN3AADRB2KDM4E
SCHEMBL8553670 0.90 SCN1A (0.61) SCN1ASCN2ASCN3AADRB2KDM4E
SCHEMBL8553837 0.89 SCN1A (0.60) SCN1ASCN2ASCN3AADRB2KDM4E
SCHEMBL8552222 0.89 SCN1A (0.60) SCN1ASCN2ASCN3AADRB2KDM4E
Hydrochloric Acid SCHEMBL27561716 0.89 SCN1A (0.60) SCN1ASCN2ASCN3AKDM4EGAA
SCHEMBL8550198 0.89 ADRB2 (0.57) ADRB2HTR2AGAA
SCHEMBL8550662 0.89 SCN1A (0.63) SCN1ASCN2ASCN3AGAA
SCHEMBL8551383 0.89 CARM1 (0.60) SCN1ASCN2ASCN3AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed