SCHEMBL8551682

SCHEMBL8551682

CC1(c2cccc(Br)c2)OCCO1.O=CCc1cccc(Br)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNB4 P30926 1/20 0.38
SLC6A4 P31645 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CHRND Q07001 1/20 0.38
HCAR3 P49019 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
TAAR1 Q96RJ0 3/20 0.35
MAOB P27338 5/20 0.35
MAOA P21397 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL855229 0.84 CHRNA1 (0.48) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL689563 0.77 TAAR1 (0.52) HCAR2TAAR1MAOBMAOASMN1; SMN2
SCHEMBL27652959 0.77 TSHR (0.40) HCAR3HCAR2SMN1; SMN2ALDH1A1
SCHEMBL8551681 0.75 MAOB (0.43) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL992385 0.71 CHRNA1 (0.49) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL7081105 0.70 TSHR (0.37) SLC6A2SLC6A4SLC6A3TAAR1ALDH1A1
SCHEMBL856168 0.70 ALDH1A1 (0.40) MAOBMAOASMN1; SMN2ALDH1A1TDP1
SCHEMBL6158666 0.70 TSHR (0.39) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL29793660 0.70 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1
SCHEMBL856097 0.70 OPRM1 (0.40) CHRNB4CHRNA3HCAR3HCAR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825992-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-03-04 EP disclosed
WO-1996036633-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-11-21 WO disclosed