SCHEMBL8551917

SCHEMBL8551917

CC(C)(C)OC(=O)N1CCC(c2cc(-c3ccc4c(c3)OCCO4)on2)CC1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCD5 Q86SK9 7/20 0.62
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
MAPT P10636 8/20 0.49
TP53 P04637 4/20 0.48
THRB P10828 2/20 0.48
LMNA P02545 2/20 0.47
MMP13 P45452 1/20 0.47
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657527 0.85 SCD5 (0.53) SCD5MAPTTP53THRBLMNA
SCHEMBL20676587 0.82 SCD5 (0.48) SCD5MAPTTHRBHTT
SCHEMBL13940704 0.81 NPC1 (0.52) SCD5NPC1RAB9AMAPTTP53
SCHEMBL20676584 0.79 SCD5 (0.45) SCD5MAPTTHRBHTT
SCHEMBL3068961 0.77 SCD5 (0.56) SCD5MAPTTP53THRBLMNA
SCHEMBL21536288 0.77 SCD5 (1.00) SCD5NPC1RAB9AMAPTTP53
SCHEMBL20676330 0.76 GPR119 (0.49) SCD5HTT
SCHEMBL12580569 0.76 SCD5 (0.59) SCD5MAPTTP53LMNAMMP13
SCHEMBL30182200 0.76 MAPT (0.49) NPC1RAB9AMAPTTHRBHTT
SCHEMBL20676655 0.75 GPR119 (0.43) SCD5MAPTTHRBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0822814-A4 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1998-12-09 EP disclosed
EP-0822814-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-02-11 EP disclosed
US-5668148-A BENIGN PROSTATIC HYPERTROPHY MERCK & CO., INC. (US) 1997-09-16 US disclosed
WO-1996032938-A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1996-10-24 WO disclosed