SCHEMBL8551930

SCHEMBL8551930

N=C(N)Nc1nnc(-c2ccccc2)c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.51
KDM4E B2RXH2 2/20 0.51
THRB P10828 1/20 0.51
ENPP3 O14638 1/20 0.48
GAA P10253 2/20 0.48
ALDH1A1 P00352 4/20 0.47
HPGD P15428 3/20 0.47
MAPT P10636 3/20 0.47
PDE5A O76074 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
CYP2C19 P33261 1/20 0.47
PDE1A P54750 1/20 0.47
PDE1B Q01064 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE1C Q14123 1/20 0.47
PDE3A Q14432 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8550943 0.98 NPSR1 (0.50) NPSR1KDM4ETHRBENPP3GAA
SCHEMBL8547920 0.88 ALDH1A1 (0.64) NPSR1THRBENPP3GAAALDH1A1
SCHEMBL8547080 0.84 KDR (0.43) NPSR1KDM4ETHRBENPP3GAA
Hydrochloric Acid SCHEMBL8549048 0.83 MEN1 (0.60) NPSR1THRBENPP3ALDH1A1HPGD
Hydrochloric Acid SCHEMBL8549372 0.82 NPSR1 (0.39) NPSR1KDM4ETHRBENPP3GAA
SCHEMBL8374822 0.82 NPSR1 (0.39) NPSR1KDM4ETHRBENPP3GAA
SCHEMBL8518196 0.82 NPSR1 (0.39) NPSR1KDM4ETHRBENPP3GAA
Hydrochloric Acid SCHEMBL8547922 0.81 NPSR1 (0.39) NPSR1KDM4ETHRBENPP3GAA
Hydrochloric Acid SCHEMBL8548606 0.81 ALDH1A1 (0.42) NPSR1KDM4ETHRBENPP3GAA
Hydrochloric Acid SCHEMBL8547376 0.81 NPSR1 (0.39) NPSR1KDM4ETHRBENPP3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed