SCHEMBL8518196

SCHEMBL8518196

N=C(N)Nc1nnc(-c2ccccc2)c2cccc(I)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.39
KDM4E B2RXH2 2/20 0.39
THRB P10828 1/20 0.39
ALDH1A1 P00352 3/20 0.38
MAPT P10636 2/20 0.38
PDE5A O76074 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDE1A P54750 1/20 0.38
PDE1B Q01064 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE1C Q14123 1/20 0.38
PDE3A Q14432 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8547922 0.99 NPSR1 (0.39) NPSR1KDM4ETHRBALDH1A1MAPT
SCHEMBL8548358 0.89 ALDH1A1 (0.46) NPSR1THRBALDH1A1MAPTHPGD
SCHEMBL8546406 0.89 SMN1; SMN2 (0.36) NPSR1KDM4ETHRBALDH1A1MAPT
SCHEMBL8374822 0.84 NPSR1 (0.39) NPSR1KDM4ETHRBALDH1A1MAPT
Hydrochloric Acid SCHEMBL8549372 0.84 NPSR1 (0.39) NPSR1KDM4ETHRBALDH1A1MAPT
Hydrochloric Acid SCHEMBL8548606 0.83 ALDH1A1 (0.42) NPSR1KDM4ETHRBALDH1A1MAPT
Hydrochloric Acid SCHEMBL8547376 0.83 NPSR1 (0.39) NPSR1KDM4ETHRBALDH1A1MAPT
SCHEMBL8518058 0.83 ADORA2A (0.36) ALDH1A1CYP1A2CYP3A4CYP2D6ALOX15
Hydrochloric Acid SCHEMBL8546924 0.82 ADORA2A (0.36) KDRSIGMAR1
SCHEMBL8551930 0.82 NPSR1 (0.51) NPSR1KDM4ETHRBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950418-A2 Composition for preventing or treating ischemic disease Takeda Chemical Industries, Ltd. (JP) 1999-10-20 EP disclosed
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed