SCHEMBL8552045

SCHEMBL8552045

Cc1c(C(F)(F)F)nn(C)c1-c1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.54
PTGS2 P35354 3/20 0.54
GRM5 P41594 4/20 0.45
CNR1 P21554 1/20 0.43
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996602 0.78 CNR1 (0.48) GRM5CNR1NR1H2NR1H3MEN1
SCHEMBL14996603 0.78 CNR1 (0.48) GRM5CNR1NR1H2NR1H3MEN1
SCHEMBL27945254 0.75 CNR1 (0.49) GRM5CNR1NR1H2NR1H3MEN1
SCHEMBL20074757 0.75 CNR1 (0.46) GRM5CNR1NR1H2NR1H3MEN1
SCHEMBL8549963 0.74 SLC34A1 (0.39) PTGS1PTGS2CNR1NR1H2NR1H3
SCHEMBL13066524 0.74 MEN1 (0.46) PTGS1PTGS2GRM5CNR1NR1H2
SCHEMBL12856425 0.74 GRM5 (0.47) GRM5CNR1NR1H2NR1H3KDM4E
SCHEMBL13066522 0.74 SMN1; SMN2 (0.46) PTGS1PTGS2GRM5NR1H2NR1H3
SCHEMBL13430367 0.72 POLB (0.54) PTGS1PTGS2NR1H2NR1H3KDM4E
SCHEMBL6013971 0.71 PTGS2 (1.00) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0846105-A1 HERBICIDAL SUBSTITUTED 3-ARYL-PYRAZOLES MONSANTO COMPANY (US) 1998-06-10 EP disclosed
US-5675017-A REACTING VINY ETHER DERIVATIVE WITH HYDRZINE OR SUBSTITUTED HYDRAZINE TO FORM A CHEMICAL INTERMEDIATE, REACTING INTERMEDIATE WITH SUBSTITUTED HALIDE OR DIALKYL SULFATE MONSANTO COMPANY (US) 1997-10-07 US disclosed
US-5672715-A Herbicidal substituted 3-aryl-pyrazoles MONSANTO COMPANY (US) 1997-09-30 US disclosed
US-5668088-A Herbicidal substituted 3-aryl-pyrazoles MONSANTO COMPANY (US) 1997-09-16 US disclosed
WO-1996040643-A1 HERBICIDAL SUBSTITUTED 3-ARYL-PYRAZOLES MONSANTO COMPANY (US) 1996-12-19 WO disclosed